MAGL INHIBITORS Russian patent published in 2021 - IPC C07D295/205 A61K31/495 A61P25/00 A61P29/00 

Abstract RU 2754536 C1

FIELD: pharmaceutics.

SUBSTANCE: invention relates to piperazine compounds of the formula (I).

EFFECT: new compounds of the formula (I) are obtained that can be used as MAGL modulators.

6 cl

Similar patents RU2754536C1

Title Year Author Number
SPIROCYCLIC COMPOUNDS AND METHODS FOR THEIR PRODUCTION AND USE 2018
  • Grajs, Sheril A.
  • Veber, Oliviya D.
  • Buzard, Deniel Dzh.
  • Shagkhafaj, Majkl B.
  • Dzhouns, Todd K.
RU2781639C2
PYRAZOLE-BASED MAGL INHIBITORS 2018
  • Grajs, Sheril A.
  • Viner, Dzhon Dzh.M.
  • Veber, Oliviya D.
  • Dunkan Katarina K.
RU2789157C2
TRANSGLUTAMINASE 2 (TG2) INHIBITORS 2019
  • Campbell, David
  • Chapman, Justin
  • Cheung, Mui, H.
  • Diraimondo, Thomas, R.
  • Duron, Sergio, G.
RU2781370C2
HETEROCYCLIC SPIRO COMPOUNDS AS MAGL INHIBITORS 2018
  • Brodney, Michael Aaron
  • Butler, Christopher Ryan
  • Helal, Christopher John
  • Mcallister, Laura Ann
  • O'Neil, Steven Victor
  • Verhoest, Patrick Robert
RU2726631C1
HETEROCYCLIC IMMUNOMODULATORS AS INHIBITOR OF IMMUNE RESPONSE CHECKPOINTS PDL1 2020
  • Mak Gouen, Devid Krejg
  • Yakobi, Edgar
RU2824127C2
11,13-MODIFIED SAXITOXINS FOR PAIN TREATMENT 2018
  • Mulkakhi, Dzhon
  • Padzhoukhesh, Khassan
  • Milanich, Dzhordzh
  • Delvig, Anton
  • Bekli, Dzhejkob
  • Shibuja, Grant Masaaki
  • Dyu Bua, Dzhastin
RU2778455C2
ROUTES OF APPLICATION OF PHOSPHODIESTERASE INHIBITORS 2020
  • Sheng, Zejuan
  • Wu, Frank
RU2795503C2
MACROCYCLIC PHENYLCARBAMATES INHIBITING HCV 2008
  • Rabuasson P'Er Zhan-Mari Bernar
  • Antonov Dmitrij
  • Ajesa Alvares Susana
  • Bel'Frage Anna Karin Gertrud Linnea
  • Jensson Karl Ehrik Daniehl'
  • Mak Govan Dehvid Krejg
  • Nil'Sson Karl Magnus
  • Rosenkvist Osa Annika Kristina
  • Samuehl'Sson Bengt Bertil'
RU2490261C2
CRYSTALLINE FORMS OF MAGL INHIBITOR 2017
  • Grajs, Sheril A.
  • Dzhons, Todd K.
  • Grimm, Kurt Dzh.
  • Blankman, Zhaklin Lorejn
  • Bils, Chenning Rodni
RU2799564C2
ROR-GAMMA MODULATORS 2017
  • Mohan, Raju
  • Nuss, Dzhon
  • Kharris, Dzheison
RU2753490C2

RU 2 754 536 C1

Authors

Grice, Cheryl A.

Buzard, Daniel J.

Shaghafi, Michael B.

Dates

2021-09-03Published

2017-11-15Filed