ORGANIC COMPOUNDS Russian patent published in 2013 - IPC A61K9/14 A61K31/40 A61K31/4412 A61P11/00 

Abstract RU 2496479 C2

FIELD: medicine, pharmaceutics.

SUBSTANCE: invention refers to a method for preparing an inhaled fine or crystalline glycopyrronium powder salt. The declared method involves suspending the crystalline glycopyrronium salt in acetone to prepare a suspension, homogenising the suspension at pressure 500-2000 bar to prepare glycopyrronium salt particles at average particle size less than 10 mcm, and drying the glycopyrronium salt particles to remove residual acetone if any.

EFFECT: invention provides preparing the aggregation and agglomeration resistant crystalline glycopyrronium powder salt.

7 cl, 2 tbl, 4 ex

Similar patents RU2496479C2

Title Year Author Number
ORGANIC COMPOUNDS 2008
  • Murer Gerkhard
  • Razenak Norbert
  • Junke Mikhaehl'
RU2482838C2
DEAMORPHIZATION OF SPRAY-DRIED FORMULATIONS VIA SPRAY-BLENDING 2014
  • Virz Dzheffri
  • Khuang Deniel
  • Tarara Tomas
  • Miller Denfort
RU2698331C2
PARTICLE SIZE REDUCTION OF ANTIMUSCARINIC COMPOUND 2014
  • Paskuali Irene
  • Kazatstsa Andrea
  • Sonders Mark
  • Lozi Elena
RU2667636C2
DRY POWDER COMPOSITIONS REPRESENTED AS PARTICLES WHICH CONTAIN TWO OR MORE ACTIVE INGREDIENTS FOR TREATMENT OF OBSTRUCTIVE OR INFLAMMATORY DISEASES OF RESPIRATORY WAYS 2012
  • Virz Dzheffri
  • Khuang Deniel
  • Miller Denfort
  • Rao Nagaradzha
  • Tarara Tomas E.
RU2629333C2
PHARMACEUTIC COMPOSITIONS 2005
  • Morton Dehvid
  • Shott Martin
  • Dehjvis Rebekka
RU2396943C2
OBTAINING MICRONIZED GLYCOPYRRONIUM SALT PARTICLES BY HYDRODYNAMIC CAVITATION 2017
  • Davanzo, Stephen P
  • Nall, Barry E
  • Rouse, Timothy J
  • Miozzi, Michele
RU2723549C2
INHALATION COMPOSITIONS CONTAINING GLYCOPYRRONIUM SALTS 2007
  • Khehberlin Barbara
  • Shtovasser Frank
  • Virt Vol'Fgang
  • Baumberger Anton
  • Abel' Shtefan
  • Kehrger Zebastian
  • Kikbush Tomas
RU2453302C2
COMPOSITIONS, METHODS AND SYSTEMS FOR RESPIRATORY DELIVERY OF TWO OR MORE ACTIVE AGENTS 2010
  • Vekhring Rejnkhard
  • Khartman Majkl Stiven
  • Smit Adrian Edvard
  • Dzhoshi Vidiya B.
  • Dvivedi Sarvadzhna Kumar
  • Lechuga-Ballesteros Devid
RU2586297C2
PHARMACEUTICAL COMPOSITIONS 2005
  • Murer Gerkhard
  • Shneeberger Rikardo
  • Virt Vol'Fgang
  • Baumberger Anton
RU2412686C2
METHOD OF PRODUCING PYRROLIDINIUM SALTS 2010
  • Tomas All'Mendinger
RU2554878C2

RU 2 496 479 C2

Authors

Murer Gerkhard

Kikbush Tomas

Singkh Dilradzh

Takur Randzhit

Shaffljuttsel' Kurt

Razenak Norbert

Dates

2013-10-27Published

2008-12-11Filed