NEW SIGMA (Σ)-RECEPTOR LIGANDS WITH ANTIAPOPTOTIC AND/OR PROAPOPTOTIC PROPERTIES IN RELATION TO BIOCHEMICAL MECHANISMS OF CELL, POSSESSING NEUROPROTECTIVE, ANTICANCER, ANTIMETASTATIC AND ANTI-INFLAMMATORY ACTION IN CHRONIC INFLAMMATORY PROCESS Russian patent published in 2013 - IPC A61K31/135 A61K31/341 A61P25/00 A61P35/00 A61P37/00 

Abstract RU 2497511 C2

FIELD: medicine, pharmaceutics.

SUBSTANCE: present invention refers to selective sigma-receptor ligands possessing prototypical biphase, antiapoptotic and proapoptotic activity in relation to normal neuronal and cancer cells, to a pharmaceutical composition based thereon, and to using the same for preparing the respective pharmaceutical products.

EFFECT: preparing the pharmaceutical products with anticancer, antimetastatic, anti-inflammatory, neuroprotective, anticonvulsant, antidepressive and nootropic analeptic or sedative action.

4 cl

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RU 2 497 511 C2

Authors

Vamvakides Aleksandr

Dates

2013-11-10Published

2008-01-14Filed