BIODEGRADABLE POLYMER CARRIER FOR ANTI-CANCER DRUG DELIVERY (VERSIONS) Russian patent published in 2013 - IPC A61K47/34 A61K47/48 C08G69/02 A61K31/335 A61P35/00 

Abstract RU 2500428 C1

FIELD: medicine, pharmaceutics.

SUBSTANCE: invention refers to medicine and describes biodegradable polymer carriers for delivery of anti-cancer drugs, particularly taxane and anthracycline antibiotic compounds. The biodegradable polymer carrier represents a polymer with its macromolecular structure being L-lysine fragments and asparaginic acid β-hydrazide and/or glutamic acid γ-hydrazide fragments. The L-lysine fragments form a linear polymer chain, while the asparaginic acid β-hydrazide and/or glutamic acid γ-hydrazide fragments form linear polymer chains with the latter being engrafted to L-lysine έ -amino groups.

EFFECT: biodegradable polymer carrier is able to bind to an anti-cancer drug to form degradable bonds in human physiologic environments.

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RU 2 500 428 C1

Authors

Vlasov Gennadij Petrovich

Paltuev Ruslan Malikovich

Semiglazov Vladimir Fedorovich

Dates

2013-12-10Published

2012-06-14Filed