METHOD OF PRODUCING NAPHTHALEN-2-YL-PYRAZOL-3-ONE INTERMEDIATE COMPOUNDS USED IN SYNTHESIS OF SIGMA RECEPTOR INHIBITORS Russian patent published in 2014 - IPC C07D231/20 

Abstract RU 2509763 C2

FIELD: chemistry.

SUBSTANCE: invention relates to novel naphthalen-2-yl-pyrazol-3-one intermediate compounds of formula (V) or (Va), a method for production thereof and use of said intermediate compounds to produce sigma receptor inhibitors.

,

where R1 denotes hydrogen, C1-6alkyl or -C(=O)R4; R2 denotes hydrogen, C1-6alkyl or phenyl; R3 denotes hydrogen or C1-6alkoxy; and R4 denotes hydrogen or C1-4alkyl.

EFFECT: obtaining novel naphthalen-2-yl-pyrazol-3-one intermediate compounds of formula (V) or (Va).

15 cl, 1 tbl, 3 ex

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RU 2 509 763 C2

Authors

Torrens Khover Antoni

Korbera Arkhona Khordi

Kuberes-Altisent Marija Rosa

Dates

2014-03-20Published

2009-04-24Filed