5-AMINO-2-(1-HYDROXYETHYL)TETRAHYDROPYRAN DERIVATIVES Russian patent published in 2014 - IPC C07D491/56 C07D497/04 C07D519/00 A61K31/4375 A61K31/498 A61P31/04 

Abstract RU 2525541 C2

FIELD: chemistry.

SUBSTANCE: invention relates to antibacterial compounds of formula

,

where R1 is an alkoxy group; R2 is H or F; each of R3, R4, R5 and R6 is independently H or D; V is CH and W is CH or N, or V is N and W is CH; Y is CH or N; Z is O, S or CH2 and A is CH2, CH2CH2 or CD2CD2; or a salt of said compound. The invention also describes a antibacterial pharmaceutical composition which contains the compound of formula (I) as a basic component, and use of the compound of formula (I).

EFFECT: obtaining novel compounds possessing useful biological properties.

25 cl, 2 tbl, 24 ex

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RU 2 525 541 C2

Authors

Kristian Khubshverlen

Georg Rjuehdi

Zhan-Filipp Sjurive

Kornelia Tsumbrunn-Aklin

Dates

2014-08-20Published

2009-12-11Filed