2-HYDROXYETHYL-1H-QUINOLIN-2-ONE DERIVATIVES AND THEIR AZAISOSTERIC ANALOGUES WITH ANTIBACTERIAL ACTIVITY Russian patent published in 2015 - IPC C07D491/56 C07D497/04 A61K31/436 A61K31/4365 A61K31/498 A61K31/4985 A61P31/04 

Abstract RU 2540862 C2

FIELD: medicine, pharmaceutics.

SUBSTANCE: invention refers to compounds of formula and their pharmaceutically acceptable salts possessing antibacterial properties, as well as to a based pharmaceutical composition. In formula (I) R1 represents an alkoxy group; each of U and V represents CH, and W represents N, or U represents N, V represents CH and W represents CH or N, or each of U and V represents N, and W represents CH; R2 represents hydrogen or fluorine, if W represents CH, or R2 represents hydrogen, if W represents N; A represents O or CH2; Y represents CH or N; Q represents O or S; and n represents 0 or 1.

EFFECT: preparing the pharmaceutically acceptable salts possessing the antibacterial properties.

23 cl, 3 tbl, 15 ex

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RU 2 540 862 C2

Authors

Kristian Khubshverlen

Georg Rjuehdi

Zhan-Filipp Sjurive

Kornelija Tsumbrunn-Aklen

Dates

2015-02-10Published

2010-04-08Filed