CRYSTALLINE FORMS OF SAXAGLIPTIN Russian patent published in 2015 - IPC C07D209/52 A61K31/403 A61P3/10 

Abstract RU 2539590 C2

FIELD: chemistry.

SUBSTANCE: invention refers to new anhydrous crystalline forms of saxagliptin hydrochloride of formula presented below There are described methods for producing the crystalline forms of saxagliptin hydrochloride.

EFFECT: crystalline forms of saxagliptin inhibit dipeptidylpeptidase-4.

13 cl, 4 tbl, 11 dwg, 5 ex

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RU 2 539 590 C2

Authors

Artur Pikhler

Jozef Vizer

Kristof Langes

Militsa Vukitsevits

Dates

2015-01-20Published

2010-04-09Filed