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2 543 375

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C1

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IPC

C07D239/60(2006-01-01)

C07C229/64(2006-01-01)

A61P29/00(2006-01-01)

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Application

2013135609/04, 2013-07-29

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Start date

2013-07-29

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Actual filing date

2013-07-29

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Published

2015-02-27

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Inventor

Borisova Natal'Ja SergeevnaZimin Jurij StepanovichGimadieva Al'Fija RaisovnaMustafin Akhat Gaziz'JanovichLarionov Sergej LeonidovichSafarova Irina Vladimirovna

(73)

Holder

Federal'Noe Gosudarstvennoe Bjudzhetnoe Obrazovatel'Noe Uchrezhdenie Vysshego Professional'Nogo Obrazovanija Gosudarstvennyj Universitet"

METHYLURACIL DERIVATIVE AND ORGANIC ACID COMPLEX AND METHOD FOR PRODUCTION THEREOF Russian patent published in 2015 - IPC C07D239/60 C07C229/64 A61P29/00 

Abstract RU 2543375 C1

FIELD: chemistry.

SUBSTANCE: invention relates to a novel complex of 5-hydroxy-6-methyluracil with 5-aminosalicylic acid of formula . The compound has anti-inflammatory activity and can be used as a basic active substance when producing novel medicinal preparations having anti-inflammatory action. The invention also relates to a method of obtaining said complex. The method includes reacting 5-hydroxy-6-methyluracil with 5-aminosalicylic acid in equimolar amounts in an aqueous medium at room temperature for 24 hours, followed by removal of water from the reaction mixture and obtaining the product.

EFFECT: wider range of pharmacological preparations with low toxicity, having higher anti-inflammatory activity.

2 cl, 1 tbl, 1 ex

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RU 2 543 375 C1

Authors

Borisova Natal'Ja Sergeevna

Zimin Jurij Stepanovich

Gimadieva Al'Fija Raisovna

Mustafin Akhat Gaziz'Janovich

Larionov Sergej Leonidovich

Safarova Irina Vladimirovna

Dates

2015-02-27—Published

2013-07-29—Filed

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