FIELD: biotechnology.
SUBSTANCE: invention relates to the field of antiparasitic agents, namely to the previously unknown insecticidal agent, which is a compound - 5-O-succinoylivermectin of formula 1, which can be used in medicine, veterinary medicine as well as agriculture, fishing industry and in other fields associated with breeding of animals, as a component for insecticides. This compound is obtained by interaction of ivermectin B with succinic anhydride in the medium of an organic solvent such as in pyridine, or in a mixture of dimethylformamide and pyridine, in the presence of a catalyst of amine type, such as for example triethylamine, dimethylaminopyridine.
EFFECT: creation of a new highly effective insecticidal agent, which is 5-O-succinoylivermectin of formula I, resistant to the action of sunlight, which then can be used to control insects in lower concentrations.
1 tbl, 3 ex
| Title | Year | Author | Number |
|---|---|---|---|
| ANTIPARASITIC AGENT | 2014 |
|
RU2554074C1 |
| 5-O-DERIVATIVES OF AVERMECTIN, METHOD FOR PRODUCTION THEREOF AND ANTIPARASITIC AGENTS BASED THEREON | 2011 |
|
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|
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| 4"-O,5-O-DI(METHYLCARBAMATE)IVERMECTIN, METHOD OF ITS PRODUCTION AND ANTIPARASITIC AGENT BASED THEREON | 2016 |
|
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| PREPARATION FOR COMBATING WITH INSECTS-CERATOPHAGES | 2016 |
|
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| METHOD OF DISINSECTION OF LIVESTOCK BUILDINGS | 2011 |
|
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| AVERMECTIN B 5-O-SUCCINATE, METHOD FOR PRODUCTION THEREOF AND ANTI-PARASITIC AGENT BASED THEREON | 2017 |
|
RU2670092C1 |
| METHOD FOR FIGHTING FLIES | 2016 |
|
RU2628936C1 |
| METHOD OF DESINSECTION OF LIVESTOCK HOUSES AND INSECTICIDAL COMPOSITION FOR ITS IMPLEMENTATION | 2011 |
|
RU2475024C2 |
| IVERMECTIN 5,4"-BIS[(ARYL)AMINO](THIOXO)ACETATES, METHOD FOR PRODUCTION THEREOF AND ANTIPARASITIC AGENTS BASED THEREON | 2017 |
|
RU2670202C1 |
