NEW OXAZOLIDINONE DERIVATIVES, METHOD FOR PRODUCING AND USING THEM Russian patent published in 2015 - IPC C07D413/14 A61K31/4439 A61P31/04

Abstract RU 2559620 C2

FIELD: medicine, pharmaceutics.

SUBSTANCE: invention refers to oxazolidinone derivatives of formula

(I),

wherein R₁ and R'₁ independently mean hydrogen or fluorine; R₂ means -OR₇, a monophosphate or a phosphate metal salt; R₇ means hydrogen or an acylated amino acid group, wherein amino acid is alanine, glycine, proline, β-alanine or valine; Het means oxadiazolyl; R₃ means C_1-4alkyl. Besides, the invention refers to a pharmaceutical composition, using it and methods for producing compounds of formula (I).

EFFECT: oxazolidinone derivatives of formula (I) possessing antibacterial activity.

28 cl, 4 tbl, 73 ex

Similar patents RU2559620C2

Title	Year	Author	Number
NOVEL OXAZOLIDINONE DERIVATIVES	2004	Rkhi Dzhae Keol Im Veon Bin Cho Chong Khvan Choj Sung Khak Li Tae Kho	RU2414469C2
NOVEL OXADIAZOLE-BASED COMPOUNDS FOR CONTROLLING PHYTOPATHOGENIC FUNGI OR PREVENTING DAMAGE BY THEM	2020	Bhujade, Paras Raybhan Naik, Maruti N Pawar, Rajesh Belkar, Yogesh Kashiram Autkar, Santosh Shridhar Garg, Ruchi Gade, Vishwanath Klausener, Alexander G.M. Kulkarni, Shantanu Ganesh Rathore, Karan	RU2818085C2
USE OF 1H-PYRAZOLO[4,3-B]PYRIDINES AS PDE1 INHIBITORS	2017	Keler, Yan Dzhukhl, Karsten Marigo, Mauro Vital, Paulo, Khorkhe, Viejra Dzhessing, Mikkel Langgard, Morten Rasmussen, Lars, Kin Klementson, Karl, Martin, Sebastian	RU2759380C2
PHENICOL ANTIBACTERIAL AGENTS	2013	Curtis Michael Duclos Brian A. Ewin Richard A. Johnson Paul D. Johnson Timothy A. Vairagoundar Rajendran Billen Denis Goodwin Richard M. Haber-Stuk Andrea K. Kyne Graham M. Sheehan Susan M.K.	RU2593204C2
PIPERIDINYLPYRAZOLOPYRIMIDINONES AND USE THEREOF	2015	Ellermann Manuel Falot Gelle Kankho Grande Iolanda Khassfeld Jorma Kintsel Tom Kebberling Jokhannes Bajer Kristin Rerig Zuzanne Shpertsel Mikhael Shtampfuss Yan Majer Imke Kellnberger Maria Burkkhardt Nils Shlemmer Karl-Khajnts Shtegmann Kristian Shumakher Joakhim Verner Mattias Khajermann Jorg Khengeveld Villem Yan	RU2713937C2
HETEROCYCLIC COMPOUND AS PROTEIN KINASE INHIBITOR	2018	Lee Hyuk Woo Ji Mi Kyung Kim Seung Chan Yu Ha Na Jung Soo Yeon Park Ji-Yeon Lee Ye-Lim Lee Ho-Youl Ki So Young Kim Dongkyu Kim Myeongjoong	RU2783723C2
PIPERIDINE DERIVATIVES	2011	Baumann Karlkhajnts Flor Aleksandr Getshi Ehrvin Grin Ljuk Zholidon Siniz Knust Khenner Limberg An'Ja Luehbbers Tomas Tomas Ehndrju	RU2554353C2
BICYCLIC TETRAHYDROTHIAZEPINE DERIVATIVES USEFUL FOR TREATING NEOPLASTIC AND/OR INFECTIOUS DISEASES	2016	Ermann Monika Lametshvandtner Gyunter Amoutseg Patrisia Leoni Kraft Rassell Styuart Khanke Tomas Dzhejms Timoti Robin Dzhouns Severin Daniel Lojbner Khans Loke Puj Leng Shternberger Ina Shtyutts Anton Ver Roland Uittejker Mark	RU2730524C2
AZADECALINS CONDENSED WITH HETEROARYLKETONES - GLUCOCORTICOID RECEPTOR MODULATORS	2013	Khant Khejzel Dzhonson Toni Rej Nikolas Uolters Ajejn	RU2639867C2
SUBSTITUTED PHENOXY-ACETIC ACIDS, WITH MODULATING EFFECT ON CRTh2 RECEPTORS	2004	Bonnert Rodzher Braf Stiven Dehvis Ehndrju Ljuker Timoti Makinalli Tomas Millichip Ajan Pehrodo Garri Pehtel Ehnil Rasul Raksana Tom Stiven	RU2372330C2

RU 2 559 620 C2

Authors

Rkhi Dzhae Keol

Im Veon Bin

Cho Chong Khvan

Choj Sung Khak

Li Tae Kho

Dates

2015-08-10—Published

2004-12-17—Filed