MACROCYCLIC COMPOUNDS, APPLIED AS HISTONE DEACETYLASE INHIBITORS Russian patent published in 2015 - IPC C07K11/02 A61K38/15 A61P35/00 

Abstract RU 2565076 C2

FIELD: medicine, pharmaceutics.

SUBSTANCE: invention relates to a novel macrocyclic compound of general formula

,

possessing an inhibiting activity with respect to histone deacetylases (HDAC), a compound-containing pharmaceutical composition, and a method, applied for the treatment of diseases with compound application.

EFFECT: obtaining the compound, possessing an inhibiting activity with respect to histone deacetylases.

11 cl, 3 tbl, 9 dwg, 11 ex

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RU 2 565 076 C2

Authors

Lju Sjuehdun

Fillips Ehndrju Dzh.

Ungermannova Dana

Nasveschuk Kristofer G.

Chzhan Gan

Dates

2015-10-20Published

2011-05-26Filed