PURINE DERIVATIVES APPLICABLE FOR TREATING FAP-RELATED (FIBROBLAST ACTIVATOR PROTEIN) DISEASES Russian patent published in 2015 - IPC A61P35/00 A61K31/5025 A61K31/517 A61K31/522 A61K31/55 A61K31/5513 A61K31/553 

Abstract RU 2569749 C2

FIELD: medicine, pharmaceutics.

SUBSTANCE: invention concerns using a compound representing 1-[(4-methylquinazolin-2-yl)methyl]-3-methyl-7-(2-butyn-1-yl)-8-(3-(R)-aminopiperidin-1-yl)-xanthine or its salt for producing a pharmaceutical composition applicable for treating hyperproliferative diseases responding to FAP (fibroblast activator protein) inhibition specified in a group consisting cirrhosis, or healing wounds, treating acne and proliferative skin diseases, such as e.g. psoriasis.

EFFECT: invention refers to using the substances, which possess an inhibitory ability for treating hyperproliferative diseases.

4 cl

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RU 2 569 749 C2

Authors

Frank Khimmel'Sbakh

Mikhaehl' Mark

Mokhammad Tadejen

Leo Tomas

Dates

2015-11-27Published

2008-08-15Filed