AZA-ADAMANTANE DERIVATIVE MONOHYDRATE Russian patent published in 2016 - IPC C07D471/18 A61K31/439 A61P25/00 A61P25/28

Abstract RU 2579121 C2

FIELD: medicine, pharmaceutics.

SUBSTANCE: invention refers to pharmaceutical composition modulating activity of α7 and/or α4β2 nicotinic acetylcholine receptors, containing a crystalline monohydrate of (4s)-4-(5-phenyl-1,3,4-thiadiazol-2-yloxy)-1-azatricyclo[3.3.1.1^3,7]decane dihydrocitrate as an active ingredient.

EFFECT: using pharmaceutical composition containing a crystalline monohydrate of (4s)-4-(5-phenyl-1,3,4-thiadiazol-2-yloxy)-1-azatricyclo[3,3,1,1^3,7]decane dihydrocitrate having high stability and poor moisture absorption.

3 cl, 9 dwg, 6 ex

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RU 2 579 121 C2

Authors

Chen Shuan

Napir Dzhejms Dzh.

Chzhan Dzheff Dzh. Z.

Brekmejer Pol Dzh.

Dates

2016-03-27—Published

2011-09-21—Filed