FIELD: chemistry.
SUBSTANCE: invention relates to the novel derivatives of 2-arylbenzofurane-7-formamide of general formula where R1 and R2 each independently on each other represent hydrogen, linear or branched C1-C4-alkyl, C3-C4-cycloalkyl or substituted 5- or 6-membered heterocycle, containing oxygen or nitrogen; or R1 and R2 together with N form a non-substituted or substituted saturated 5- or 6-membered heterocycle, containing at least one heteroatom, where the heteroatom represents O, N and S, the substituent represents methyl on N; R3 represents a hydrogen atom or a chlorine atom; R4 represents a hydrogen atom or a fluorine atom; X represents CH, CF or N; and Y represents CH, CF or N, or its pharmacologically or physiologically acceptable salt, as well as to a method for obtaining thereof and application in obtaining anti-tumour and anti-inflammation medications.
EFFECT: increased efficiency of the compound application.
8 cl, 5 tbl, 24 ex
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Authors
Dates
2016-05-10—Published
2013-01-14—Filed