METHOD OF PRODUCING PHENOXYPYRIDINE DERIVATIVE Russian patent published in 2016 - IPC C07D401/14 C07D401/12 C07C231/02 A61K31/496 

Abstract RU 2590158 C2

FIELD: chemistry.

SUBSTANCE: invention relates to a method of producing a compound or salt thereof of formula (I), which involves reaction of compound or salt thereof of formula (II), and aniline derivative of formula (III), in water or a mixed solvent of water and organic solvent in presence of 1-ethyl-3-(3-dimethylaminopropyl)carbodiimide and substantially in absence of a base:

.

EFFECT: technical outcome is a novel improved method of producing a compound or salt thereof of formula (I).

3 cl, 1 tbl, 5 ex

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RU 2 590 158 C2

Authors

Takakhasi Masabumi

Dates

2016-07-10Published

2012-03-27Filed