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2 593 885

(13)

(51)

IPC

A61K31/5513(2006-01-01)

C07D243/24(2006-01-01)

A61P25/08(2006-01-01)

A61P25/22(2006-01-01)

(21) (22)

Application

2015114844/15, 2015-04-20

(24)

Start date

2015-04-20

(22)

Actual filing date

2015-04-20

(45)

Published

2016-08-10

(72)

Inventor

Bespalov Aleksandr YakovlevichMatveeva Lidiya PetrovnaPetrov Aleksandr NikolaevichSavateeva Tatyana NikolaevnaChigareva Svetlana Mikhajlovna

(73)

Holder

Federalnoe Gosudarstvennoe Byudzhetnoe Uchrezhdenie Nauki Toksikologii Federalnogo Mediko-Biologicheskogo Agentstva"

ANTICONVULSANT AND TRANQUILISING AGENT Russian patent published in 2016 - IPC A61K31/5513 C07D243/24 A61P25/08 A61P25/22

Abstract RU 2593885 C1

FIELD: pharmaceutics.

SUBSTANCE: invention refers to pharmaceutics. Described is an anticonvulsant and tranquilising agent with the general formula of:

where R=CH2CH2NH2 HBr (derivative 1); R=CH2CH2CH2NH2 HBr (derivative 2); R=CH2(CH2)4NH2 HBr (derivative 3); R=p-CH₂NEt₂ HCl (derivative 4); R=m-CH₂NEt₂ HCl (derivative 5).

EFFECT: invention provides considerable reduction of time of pharmacological effect coming, as well as reduction of negative side effects.

1 cl, 7 tbl, 9 ex

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RU 2 593 885 C1

Authors

Bespalov Aleksandr Yakovlevich

Matveeva Lidiya Petrovna

Petrov Aleksandr Nikolaevich

Savateeva Tatyana Nikolaevna

Chigareva Svetlana Mikhajlovna

Dates

2016-08-10—Published

2015-04-20—Filed