NEW POLYMORPHIC FORM OF A CALCIEMETRIC COMPOUND Russian patent published in 2016 - IPC C07C213/10 C07C217/74 C07C229/46 A61K31/196 A61P3/14 A61P5/18 

Abstract RU 2599788 C2

FIELD: chemistry.

SUBSTANCE: invention is related to a crystalline form of X {4-[(1R, 3S)-3-((R)-1-naphthalene-1-ilethylamino) cyclopentyl] phenoxy} acetic acid, which can be used for treating, relieving or preventing the physiological disorders or diseases associated with disturbed activity of CaSR, such as hyperparathyroidism. This form has x-ray powder diffraction pattern, which demonstrates characteristic peaks expressed in 2θ, equal to approximately 8.0, 11.3, 11.4, 15.0, 18.2 and/or 21.5 degrees (±0.05 degrees) (underlined is the primary).

EFFECT: invention is also related to a pharmaceutical compound containing the crystalline form of X, and methods for preparing it.

19 cl, 10 dwg, 6 tbl, 5 ex

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RU 2 599 788 C2

Authors

Ebdrup Seren

Nilsen Kim Tronsegord

Greve Tanya Mariya

Dates

2016-10-20Published

2011-06-24Filed