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(19)

(11)

2 600 983

(13)

(51)

IPC

C07D409/14(2006-01-01)

C07D409/04(2006-01-01)

C07D231/14(2006-01-01)

C07D401/14(2006-01-01)

C07D403/14(2006-01-01)

C07D413/12(2006-01-01)

C07D413/14(2006-01-01)

C07D417/14(2006-01-01)

C07D471/08(2006-01-01)

C07D487/08(2006-01-01)

A61K31/454(2006-01-01)

A61K31/496(2006-01-01)

A61K31/5377(2006-01-01)

A61K31/541(2006-01-01)

A61P3/00(2006-01-01)

A61P9/00(2006-01-01)

(21) (22)

Application

2013125232/04, 2012-09-25

(24)

Start date

2012-09-25

(22)

Actual filing date

2012-09-25

(45)

Published

2016-10-27

(72)

Inventor

Shia Kak-ShanChan Chun-PinChao Yuj-Shen

(73)

Holder

Neshnl Khelt Riserch Instityuts

PYRAZOLE DERIVATIVES Russian patent published in 2016 - IPC C07D409/14 C07D409/04 C07D231/14 C07D401/14 C07D403/14 C07D413/12 C07D413/14 C07D417/14 C07D471/08 C07D487/08 A61K31/454 A61K31/496 A61K31/5377 A61K31/541 A61P3/00 A61P9/00

Abstract RU 2600983 C2

FIELD: chemistry.

SUBSTANCE: pyrazole derivatives are disclosed, which are encompassed by formula (I), in which radicals and groups are defined in patent claim and which are suitable for treating disorders mediated by peripheral cannabinoid 1 receptor 1.

EFFECT: invention also discloses pharmaceutical compositions and methods related to use of said compounds.

29 cl, 11 ex

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RU 2 600 983 C2

Authors

Shia Kak-Shan

Chan Chun-Pin

Chao Yuj-Shen

Dates

2016-10-27—Published

2012-09-25—Filed