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(19)

(11)

2 654 213

(13)

(51)

IPC

C07D231/18(2006-01-01)

C07D333/34(2006-01-01)

C07D409/12(2006-01-01)

C07D417/12(2006-01-01)

C07D413/12(2006-01-01)

C07D405/12(2006-01-01)

C07D513/04(2006-01-01)

A61K31/343(2006-01-01)

A61K31/4436(2006-01-01)

A61K31/18(2006-01-01)

(21) (22)

Application

2013132649, 2011-12-12

(24)

Start date

2011-12-12

(22)

Actual filing date

2011-12-12

(45)

Published

2018-05-17

(72)

Inventor

Yuan KhajtsinBird Richard L.Lyu SyaosyaDonello Dzhon E.Visvanat VeenaGarst Majkl E.

(73)

Holder

Allergan, Ink.

NOVEL 1,2-BIS-SULPHONAMIDE DERIVATIVES AS MODULATORS OF CHEMOKINE RECEPTOR Russian patent published in 2018 - IPC C07D231/18 C07D333/34 C07D409/12 C07D417/12 C07D413/12 C07D405/12 C07D513/04 A61K31/343 A61K31/4436 A61K31/18

Abstract RU 2654213 C9

FIELD: chemistry.

SUBSTANCE: invention relates to novel bis-sulphonamide derivatives of formula I:

as well as to pharmaceutical compositions based thereon.

EFFECT: technical result: novel compounds are obtained, which are suitable for the treatment of inflammatory diseases of the eyes or skin inflammatory diseases.

9 cl, 2 tbl

Формула I - Formula I

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RU 2 654 213 C9

Authors

Yuan Khajtsin

Bird Richard L.

Lyu Syaosya

Donello Dzhon E.

Visvanat Veena

Garst Majkl E.

Dates

2018-05-17—Published

2011-12-12—Filed