THERAPEUTIC USE OF THE TLR AGONIST AND COMBINED THERAPY Russian patent published in 2016 - IPC A61K31/55 A61K31/40 A61K31/704 A61K35/00 

Abstract RU 2603467 C2

FIELD: medicine.

SUBSTANCE: group of inventions is related to chemotherapy. Invention discloses a method of treatment of cancer including administering a compound, that contains benzo[b]azepine agonist TLR8 2-amino-N,N-dipropil-8-(4-(pyrrolidine-1-Carbonyl)phenyl)-3H-benzo[b]azepine-4-carboxamide (VTX) or its pharmaceutically acceptable salt and pharmaceutically acceptable carrier, in combination with doxorubicin, and a kit for treatment of cancer including containers with the said connections.

EFFECT: technical result consists in synergetic suppressing of the tumor volume by the declared combination of VTX + doxorubicin.

33 cl, 2 tbl, 24 dwg

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Authors

Khershberg Robert

Kukos Dzhordzh

Ditsh Gregori

Fachchjabene Andrea

Mandzharrez Kristi

Rendall Tressa D.

Dates

2016-11-27Published

2011-10-03Filed