ESTER PRODRUGS OF [3-(1-(1H-IMIDAZOL-4-YL)ETHYL)-2-METHYLPHENYL]METHANOL Russian patent published in 2017 - IPC C07D233/64 A61K31/4174 A61P27/06 

Abstract RU 2612351 C2

FIELD: chemistry.

SUBSTANCE: invention relates to specific derivatives of [3-(1-(1H-imidazol-4-yl)ethyl)-2-methylphenyl]methanol. The invention also relates to specific intermediates, and pharmaceutical compositions based on the [3-(1-(1H-imidazol-4-yl)ethyl)-2-methylphenyl]methanol derivative.

EFFECT: new heterocyclic derivatives are obtained useful for treatment of conditions mediated by adrenergic receptors.

4 cl, 2 dwg, 3 tbl, 13 ex

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RU 2 612 351 C2

Authors

Dates

2017-03-07Published

2011-09-16Filed