HYDROHALOGENIDE OF 1-(3,4-DIMETHOXYPHENYL)-2-(7,8-DIMETHYL-2,3,4,5-TETRAHYDRO-1,3]DIAZEPINO[1,2A]BENZIMIDAZOLE-11-YL)ETHANONE WITH ANALGESIC AND ANXIOLYTIC ACTIVITY Russian patent published in 2017 - IPC C07D487/04 A61K31/551 A61P29/00 

Abstract RU 2636785 C1

FIELD: pharmacology.

SUBSTANCE: invention relates to organic chemistry, namely to a hydrohalogenide of 1-(3,4-dimethoxyphenyl)-2-(7,8-dimethyl-2,3,4,5-tetrahydro[1,3]diazepino[1,2-a]benzimidazole-11-yl)ethanone of formula 1

,

which has both analgesic and anxiolytic activity.

EFFECT: new heterocyclic compound possessing the effective biological properties is obtained.

2 cl, 3 tbl, 1 ex

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RU 2 636 785 C1

Authors

Divaeva Lyudmila Nikolaevna

Spasov Aleksandr Alekseevich

Maltsev Dmitrij Vasilevich

Kuzmenko Tatyana Andreevna

Morkovnik Anatolij Savelevich

Yakovlev Dmitrij Sergeevich

Taran Alena Sergeevna

Petrov Vladimir Ivanovich

Bogoslavtseva Mariya Vladimirovna

Dates

2017-12-01Published

2016-11-21Filed