TRICYCLIC BENZOXABORAL COMPOUND, METHOD FOR ITS PRODUCTION AND ITS APPLICATION Russian patent published in 2017 - IPC C07F5/02 A61K31/69 A61P31/04 

Abstract RU 2639153 C2

FIELD: pharmacology.

SUBSTANCE: invention relates to a new tricyclic benzoxaboral compound represented by chemical formula 1, its isomer or a pharmaceutically acceptable salt thereof. Chemical formula 1

Also, methods of preparation of the said compound and a pharmaceutical composition are provided.

EFFECT: new tricyclic benzoxaboral compound has antibiotic activity against gram-negative bacteria, including against gram-negative bacteria with multiple drug resistance.

14 cl, 3 tbl, 12 ex

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RU 2 639 153 C2

Authors

Kim Soon-Hoe

Im Weon-Bin

Ha Seung-Bum

Park Jung-Sang

Kim Mi-Yeon

Choi Sung-Hak

Sung Hyun-Jung

Dates

2017-12-20Published

2014-07-28Filed