PYRROLE SUBSTITUTED INDOLONE DERIVATIVE, METHOD OF ITS PREPARATION INCLUDING ITS COMPOSITION AND APPLICATION Russian patent published in 2018 - IPC C07D401/14 C07D403/14 A61K31/4045 A61K31/454 A61K35/00 

Abstract RU 2650682 C2

FIELD: medicine; pharmaceuticals.

SUBSTANCE: invention relates to a pyrrole substituted indolone derivative of formula (I), a pharmaceutical composition, comprising said derivative, and the use of pyrrole substituted indolone derivatives for the treatment of tyrosine kinase receptor mediated diseases, such as tumors.

.

EFFECT: for the treatment of tyrosine kinase receptor mediated diseases, such as tumors.

10 cl, 20 ex, 4 tbl

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RU 2 650 682 C2

Authors

Khu Likhun

Chzhao Shaokhua

Lyu Pen

Li Syantszyun

An Tszyunyun

Chzhou Mynsya

Chzhan Lili

Yao Tszytszyan

Dates

2018-04-17Published

2015-02-04Filed