ENZYME-ACTIVATING COMPOUNDS AND COMPOSITIONS Russian patent published in 2018 - IPC C07D295/192 C07D403/12 A61K31/495 A61P35/00 

Abstract RU 2652989 C2

FIELD: pharmaceuticals.

SUBSTANCE: invention relates to novel compounds of formula I:

, as well as pharmaceutical compositions based thereon.

EFFECT: obtaining novel compounds that activate procaspase-3, which can induce the death of cancer cells.

8 cl, 2 tbl, 3 ex, 10 dwg

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RU 2 652 989 C2

Authors

Hergenrother Paul J.

Roth Howard Steven

Dates

2018-05-04Published

2013-08-05Filed