APPLICATION OF 2,6-DIMETHYLPHENYLACETAMIDE DERIVATIVES WITH LOCAL ANESTHETIC ACTIVITY FOR INFILTRATION AND CONDUCTION ANESTHESIA Russian patent published in 2018 - IPC A61K31/5375 A61P23/02 

Abstract RU 2657613 C1

FIELD: medicine.

SUBSTANCE: invention relates to medicine. Use of 2,6-dimethylphenylacetamide-N-allyl-N-(2,6-dimethylphenylaminocarbonylmethyl) morpholinium bromide derivative of formula (1), with local anesthetic activity for infiltration and conduction local anesthesia. Invention can find application in medical practice for local anesthesia, in surgical and dental practice and can be used to create a domestic medicinal product of the intended use.

(1).

EFFECT: increase in the breadth of the therapeutic effect, depth and duration of infiltration and conduction local anesthesia in comparison with lidocaine.

1 cl, 3 tbl

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RU 2 657 613 C1

Authors

Kurganov Nikolaj Aleksandrovich

Skachilova Sofiya Yakovlevna

Blinov Dmitrij Sergeevich

Vasilkina Olga Vladimirovna

Novikov Andrej Vasilevich

Blinova Ekaterina Valerevna

Dates

2018-06-14Published

2017-08-16Filed