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2 705 591

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IPC

C07D487/04(2006-01-01)

A61K31/519(2006-01-01)

A61P31/06(2006-01-01)

(21) (22)

Application

2018129361, 2018-08-10

(24)

Start date

2018-08-10

(22)

Actual filing date

2018-08-10

(45)

Published

2019-11-11

(72)

Inventor

Krasavin Mikhail YurevichTrifonov Rostislav EvgenevichTolstyakov Vladimir VladimirovichDarin Dmitrij ViktorovichVinogradova Tatyana IvanovnaManicheva Olga AlekseevnaDogonadze Marine ZaurievnaZabolotnykh Natalya VyacheslavovnaVitovskaya Mariya LvovnaYablonskij Petr Kazimirovich

(73)

Holder

Federalnoe Gosudarstvennoe Byudzhetnoe Uchrezhdenie Nauchno-Issledovatelskij Institut Ftiziopulmonologii" Ministerstva Zdravookhraneniya Rossijskoj Federatsii

5-METHYL-7-(3-NITRO-[1,2,4]TRIAZOL-1-YL)-[1,2,4]TRIAZOLO[1,5-A]PYRIMIDINE, HAVING ANTI-TUBERCULOSIS ACTIVITY AGAINST THE AGENT WITH MULTIPLE DRUG RESISTANCE, AND A METHOD FOR PRODUCTION THEREOF Russian patent published in 2019 - IPC C07D487/04 A61K31/519 A61P31/06

Abstract RU 2705591 C1

FIELD: medicine.

SUBSTANCE: invention relates to use of 5-methyl-7-(3-nitro-[1,2,4]triazol-1-yl)-[1,2,4]triazolo[1,5-a]pyrimidine of formula 1 as an anti-tuberculosis substance with activity on a multiple drug resistance agent.

EFFECT: disclosed is use of 5-methyl-7-(3-nitro-[1,2,4]triazol-1-yl)-[1,2,4]triazolo[1,5-a]pyrimidine for treating tuberculosis with multiple drug resistance.

1 cl, 5 dwg, 4 tbl, 4 ex

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RU 2 705 591 C1

Authors

Krasavin Mikhail Yurevich

Trifonov Rostislav Evgenevich

Tolstyakov Vladimir Vladimirovich

Darin Dmitrij Viktorovich

Vinogradova Tatyana Ivanovna

Manicheva Olga Alekseevna

Dogonadze Marine Zaurievna

Zabolotnykh Natalya Vyacheslavovna

Vitovskaya Mariya Lvovna

Yablonskij Petr Kazimirovich

Dates

2019-11-11—Published

2018-08-10—Filed