DERIVATIVES OF PREGNENOLONE Russian patent published in 2018 - IPC C07J7/00 A61K31/57 A61P25/00 

Abstract RU 2667065 C2

FIELD: chemistry.

SUBSTANCE: present invention relates to the compound of Formula I, in which R1 represents C1-8 alkyl, C1-8 alkoxy, CN, COOCH3 or halogen, and R2 represents H, C1-8 alkyl, Bn-. Invention also relates to the pharmaceutical composition, to the compound of Formula I preparation method, to the human or animal body treatment method. Formula I.

EFFECT: technical result: new compounds of Formula I have been produced, which possess the CB1 receptor inhibitor properties, can be used in the human or animal treatment suffering from the associated with CB-1 pathology.

10 cl, 2 tbl

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RU 2 667 065 C2

Authors

Pyatstsa Per Vinchentso

Valle Monik

Felpen Fransua-Ksave

Reve Zhan-Mishel

Fabr Sandi

Dates

2018-09-14Published

2013-11-27Filed