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(19)

(11)

2 672 873

(13)

(51)

IPC

C07D498/04(2006-01-01)

C07D513/04(2006-01-01)

A61K31/424(2006-01-01)

A61P3/00(2006-01-01)

(21) (22)

Application

2015120556, 2013-10-30

(24)

Start date

2013-10-30

(22)

Actual filing date

2013-10-30

(45)

Published

2018-11-20

(72)

Inventor

Kaul RameshMakichern Ernest Dzh.Vokaldo Devid Dzh.Chzhou YuansiDan TsyunSelnik Garold Dzh.

(73)

Holder

Alektos Terapyutiks Ink.Merk Sharp I Doum Korp.

GLYCOSIDASE INHIBITORS AND THEIR APPLICATIONS Russian patent published in 2018 - IPC C07D498/04 C07D513/04 A61K31/424 A61P3/00

Abstract RU 2672873 C2

FIELD: pharmaceuticals; medicine.

SUBSTANCE: invention relates to compounds of formula (I) (I).

EFFECT: new compounds having inhibitory activity against O-GlcNAc, as well as pharmaceutical compositions based on them and methods for the treatment of mediated diseases are obtained.

22 cl, 2 tbl, 40 ex

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RU 2 672 873 C2

Authors

Kaul Ramesh

Makichern Ernest Dzh.

Vokaldo Devid Dzh.

Chzhou Yuansi

Dan Tsyun

Selnik Garold Dzh.

Dates

2018-11-20—Published

2013-10-30—Filed