THERAPEUTIC AND/OR PREVENTIVE AGENT COMPRISING 1-INDANSULFAMIDE DERIVATIVE FOR PAIN Russian patent published in 2019 - IPC A61K31/18 A61P25/04 

Abstract RU 2678571 C1

FIELD: medicine.

SUBSTANCE: invention relates to medicine, in particular to a therapeutic and/or preventive agent for acute and/or chronic pain. Said therapeutic and/or preventive agent contains, as its active agent, a compound based on 1-indansulfamide selected from the group: N-[(1S)-2,2,5,7-tetrafluoro-2,3-dihydro-1H-indene-1-yl]sulfamide, (-)-N-(7-chloro-2,2,5-trifluoro-2,3-dihydro-1H-indene-1-yl)sulfamide, N-[(1S)-2,2-difluoro-7-methyl-2,3-dihydro-1H-indene-1-yl]sulfamide N-[(1S)-2,2,5-trifluoro-7-methyl-2,3-dihydro-1H-indene-1-yl]sulfamide, or its pharmaceutically acceptable salt.

EFFECT: use of the invention provides an analgesic effect in various animal models and may be used for various types of pain.

5 cl, 10 tbl, 9 ex, 2 dwg

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RU 2 678 571 C1

Authors

Khigasiyama Khiroyuki

Kadzuta Yudzi

Khasimoto Keisuke

Dates

2019-01-30Published

2014-12-17Filed