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(19)

RU

(11)

2 688 159

(13)

C2

(51)

IPC

C07J17/00(2006-01-01)

C07J5/00(2006-01-01)

C07J31/00(2006-01-01)

A61K31/575(2006-01-01)

A61K31/58(2006-01-01)

A61P27/02(2006-01-01)

(21) (22)

Application

2014123472, 2012-11-09

(24)

Start date

2012-11-09

(22)

Actual filing date

2012-11-09

(45)

Published

2019-05-20

(72)

Inventor

Edelman Dzheffri L.Neme AlissarMaloun Tomas K.

(73)

Holder

Allergan, Ink.

4-PREGENEN-11Β-17-21-TRIOL-3,20-DIONE DERIVATIVES FOR TREATING EYE DISEASES Russian patent published in 2019 - IPC C07J17/00 C07J5/00 C07J31/00 A61K31/575 A61K31/58 A61P27/02 

Abstract RU 2688159 C2

FIELD: chemistry.

SUBSTANCE: invention relates to novel derivatives of formula I, as well as to pharmaceutical compositions based thereon

.

EFFECT: technical result is obtaining new compounds having agonistic activity on glucocorticoid or mineralocorticoid receptors, which can be used for treating disorders associated with modulation of glucocorticoid or mineralocorticoid receptor, for example, dry eyes.

10 cl, 3 tbl, 12 ex

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RU 2 688 159 C2

Authors

Edelman Dzheffri L.

Neme Alissar

Maloun Tomas K.

Dates

2019-05-20—Published

2012-11-09—Filed

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