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RU

(11)

2 693 457

(13)

C2

(51)

IPC

C07D211/14(2006-01-01)

C07D295/13(2006-01-01)

A61K31/495(2006-01-01)

A61K31/496(2006-01-01)

A61P25/00(2006-01-01)

(21) (22)

Application

2016101085, 2014-07-10

(24)

Start date

2014-07-10

(22)

Actual filing date

2014-07-10

(45)

Published

2019-07-03

(72)

Inventor

Bottegoni DzhovanniDe Simone AlessioRuda Dzhan FilippoKavalli AndreaBandera TitsianoPomelli Daniele

(73)

Holder

Fondatsone Istituto Italyano Di TeknolodzhiyaDze Ridzhents Of Dze Yuniversiti Of Kaliforniya

PHENYLCARBAMATES AND USE THEREOF AS ENZYME INHIBITORS OF HYDROLASES OF FATTY ACID AMIDES (FAAH) AND DOPAMINE RECEPTOR D3 (D3DR) MODULATORS Russian patent published in 2019 - IPC C07D211/14 C07D295/13 A61K31/495 A61K31/496 A61P25/00 

Abstract RU 2693457 C2

FIELD: chemistry.

SUBSTANCE: invention refers to compounds of formula (I) or their pharmaceutically acceptable salts.

EFFECT: technical result is obtaining novel compounds of formula (I), as well as pharmaceutical compositions based thereon, which are simultaneously inhibitors of the enzyme hydrolase amides of fatty acids (FAAH) and dopamine receptor (D3DR) D3 modulators, suitable for treating or preventing mediated disorders.

20 cl, 1 tbl, 45 ex

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RU 2 693 457 C2

Authors

Bottegoni Dzhovanni

De Simone Alessio

Ruda Dzhan Filippo

Kavalli Andrea

Bandera Titsiano

Pomelli Daniele

Dates

2019-07-03—Published

2014-07-10—Filed

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