FIELD: chemistry.
SUBSTANCE: invention relates to organic chemistry and specifically to a novel negative modulator of kainate receptors – 6-[4-methoxy-3-(pyrrolidin-1-ylmethyl)benzyl]-1,11-dimethyl-3,6,9-triazatricyclo [7.3.1.13,11]tetradecane-4,8,12-trion, the structure below or its pharmaceutically acceptable salt. Invention also relates to use of the compound of the given formula and to a pharmaceutical composition based thereon.
EFFECT: obtaining a novel heterocyclic compound which is a high-efficiency negative modulator of kainate receptors useful for treating psychic diseases, depressive disorders, anxiety disorders and stress-related disorders.
14 cl, 6 dwg, 1 ex
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