FIELD: medicine.
SUBSTANCE: invention relates to a PDE1 inhibitor applicable in medicine, characterized by a structure selected from:
,
,
,
,
, a pharmaceutical composition based thereon for treating and preventing the disease, CNS disorders or injuries.
EFFECT: novel effective PDE1 inhibitors with prolonged half-life in vivo are proposed for treating diseases, disorders and injures of the brain and spinal cord.
11 cl, 12 ex
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Authors
Dates
2020-01-17—Published
2015-09-17—Filed