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2 716 502

(13)

(51)

IPC

C07J63/00(2006-01-01)

A61K31/58(2006-01-01)

A61P31/18(2006-01-01)

(21) (22)

Application

2018130181, 2017-02-02

(24)

Start date

2017-02-02

(22)

Actual filing date

2017-02-02

(45)

Published

2020-03-12

(72)

Inventor

Chen JieChen YanDicker Ira B.Hartz Richard AMeanwell Nicholas ANowicka-Sans BeataRegueiro-Ren AliciaSit Sing-YuenSin NySwidorski JacobVenables Brian Lee

(73)

Holder

Viiv Healthcare Uk Limited

C-3 AND C-17 MODIFIED TRITERPENOIDS AS HIV-1 INHIBITORS Russian patent published in 2020 - IPC C07J63/00 A61K31/58 A61P31/18

Abstract RU 2716502 C2

FIELD: medicine; pharmaceuticals.

SUBSTANCE: invention refers to a compound, its diastereomers and pharmaceutically acceptable salts. Invention also relates to a pharmaceutical composition and to a method of treating a HIV-infected mammal.

EFFECT: technical result is obtaining novel compounds which are useful as HIV maturation inhibitors.

7 cl, 4 tbl, 75 ex

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RU 2 716 502 C2

Authors

Chen Jie

Chen Yan

Dicker Ira B.

Hartz Richard A

Meanwell Nicholas A

Nowicka-Sans Beata

Regueiro-Ren Alicia

Sit Sing-Yuen

Sin Ny

Swidorski Jacob

Venables Brian Lee

Dates

2020-03-12—Published

2017-02-02—Filed