SOLID FORMULATION FOR ORAL ADMINISTRATION CONTAINING IRINOTECAN, AND METHOD FOR PRODUCTION THEREOF Russian patent published in 2020 - IPC A61K9/16 A61K9/20 A61K9/48 A61K31/4745 A61K47/12 

Abstract RU 2716595 C2

FIELD: medicine.

SUBSTANCE: group of inventions relates to the field of medicine, specifically to a solid formulation for oral administration, containing moist granules containing irinotecan hydrochloride trihydrate and an acidifier, where the acidulent is selected from a group consisting of acetic acid, citric acid, lactic acid and any combinations thereof, and a method for production thereof.

EFFECT: group of inventions provides higher degree of dissolution of the active ingredient and provides improved bioavailability in oral administration.

9 cl, 3 dwg, 8 tbl, 6 ex

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RU 2 716 595 C2

Authors

Park Caleb Hyung Min

Jung Myeong Ki

Kim Jin Cheul

Kim Yong Il

Park Jae Hyun

Woo Jong Soo

Dates

2020-03-13Published

2016-06-20Filed