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2 719 583

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IPC

C07D487/04(2006-01-01)

(21) (22)

Application

2016151208, 2015-05-28

(24)

Start date

2015-05-28

(22)

Actual filing date

2015-05-28

(45)

Published

2020-04-21

(72)

Inventor

Akhmad NadiyaSharrer Zhan-DamenDevis KrisEtksebarriya I Khardi GorkaFrajss DamenNegtel RonaldPanesar ManinderPerar FransuazPinder DzhoannStork Per-AnriStadli Dzhon

(73)

Holder

Verteks Farmasyutikalz Inkorporejted

RADIOLABELLED 2-AMINO-6-FLUORO-N-[5-FLUORO-PYRIDIN-3-YL]-PYRAZOLO [1, 5-A] PYRIMIDINE-3-CARBOXAMIDE DERIVATIVES USED AS ATR KINASE INHIBITOR, PREPARATIONS BASED THEREON COMPOUNDS AND VARIOUS SOLID FORMS THEREOF Russian patent published in 2020 - IPC C07D487/04

Abstract RU 2719583 C2

FIELD: chemistry.

SUBSTANCE: present invention relates to a method of producing a compound of formula I-1, which includes a step of reacting a compound of formula 6b with a compound of formula 11.

EFFECT: said compound is suitable as an ATR protein kinase inhibitor.

10 cl, 9 dwg, 6 tbl, 8 ex

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RU 2 719 583 C2

Authors

Akhmad Nadiya

Sharrer Zhan-Damen

Devis Kris

Etksebarriya I Khardi Gorka

Frajss Damen

Negtel Ronald

Panesar Maninder

Perar Fransuaz

Pinder Dzhoann

Stork Per-Anri

Stadli Dzhon

Dates

2020-04-21—Published

2015-05-28—Filed