NOVEL COMPOUNDS FOR DIAGNOSING, TREATING AND PREVENTING DISEASES ASSOCIATED WITH ALPHA-SYNUCLEIN AGGREGATION Russian patent published in 2024 - IPC C07D401/04 C07D401/14 C07D403/04 C07D405/14 A61K31/4439 A61K31/444 A61K31/506 A61P25/16 A61P25/28 

Abstract RU 2822486 C1

FIELD: chemistry.

SUBSTANCE: invention relates to compounds of general formulas Ia, Ib, IIa or IIb:

,

a pharmaceutical composition based thereon, as well as the use and method of imaging alpha-synuclein and for diagnosing diseases which are associated with alpha-synuclein aggregation.

EFFECT: obtaining novel compounds which are suitable for treating and preventing diseases associated with alpha-synuclein aggregation.

20 cl, 5 ex, 7 tbl, 1 dwg

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RU 2 822 486 C1

Authors

Giese, Armin

Schmidt, Felix

Weckbecker, Daniel

Leonov, Andrei

Ryazanov, Sergey

Griesinger, Christian

Pichler, Bernd

Herfert, Kristina

Maurer, Andreas

Kuebler, Laura

Buss, Sabrina

Dates

2024-07-08Published

2020-11-19Filed