SUBSTITUTED AMINO SIX-MEMBER SATURATED HETEROALICYCLES AS LONG-ACTING DPP-IV INHIBITORS Russian patent published in 2020 - IPC C07D513/14 C07D487/04 C07D495/04 C07D405/04 A61K31/4035 A61K31/407 A61K31/4162 A61K31/542 A61P3/10 A61P5/50 

Abstract RU 2720488 C2

FIELD: medicine; pharmaceuticals.

SUBSTANCE: invention refers to compounds of formula (V), a pharmaceutical composition, as well as to application in treatment of disease and/or prevention of diseases and disorders, in which inhibition of DPP-IV is beneficial.

EFFECT: obtaining novel compounds of formula (V), having DPP-IV inhibitor activity.

8 cl, 2 dwg, 6 tbl, 9 ex

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RU 2 720 488 C2

Authors

Xu, Xinhe

Shen, Yu

Xiao, Dengming

Luo, Hong

Peng, Yong

Han, Yongxin

Zhang, Aiming

Yang, Ling

Dates

2020-04-30Published

2016-02-04Filed