AMINE COMPOUNDS HAVING ANTI-INFLAMMATORY, ANTIFUNGAL, ANTI-PARASITIC AND ANTICANCER ACTIVITY Russian patent published in 2020 - IPC C07D239/94 A61K31/517 A61P29/00 A61P31/10 A61P35/00 

Abstract RU 2721418 C2

FIELD: chemistry.

SUBSTANCE: invention relates to organic chemistry and specifically to a heterocyclic compound of formula IB1 or a pharmaceutically acceptable salt thereof, where n = 1; Q is absent; R1 denotes hydrogen; and R7 denotes phenyl substituted with alkoxy having 6–10 carbon atoms or phenoxy. Invention also relates to a method of treatment or prevention based on using the compound of formula IA1a, use of the compound of formula IB1 and composition based thereon.

EFFECT: technical result is obtaining novel heterocyclic compounds useful in treating an inflammatory disease, fungal infection, unicellular parasitic infection and tumour disease.

36 cl, 41 tbl, 171 ex

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RU 2 721 418 C2

Authors

Simpson, Devid, M.

Zerbi, Dennis, Brajan

Lu, Min

Von Borstel, Rejd, V.

Li, Zhuj

Riding, Dzhilian

Uolp, Stefen

Aman, Nureddin

Dates

2020-05-19Published

2014-01-31Filed