AMIDE (E)-2-AMINO-4-OXO-5-(2-OXO-2-PHENYLETHYLIDENE)-1-(3-ETHOXYCARBONYL)-4,5,6-7-TETRAHYDROBENZO[B]THIOPHEN-2-YL)4,5-DIHYDRO-1H-PYRROLE-3-CARBOXYLIC ACID, HAVING ANTIMICROBIAL ACTIVITY Russian patent published in 2020 - IPC C07D409/04 A61K31/38 A61K31/40 A61P31/04 

Abstract RU 2738405 C1

FIELD: chemistry.

SUBSTANCE: invention relates to amide (E)-2-amino-4-oxo-5-(2-oxo-2-phenylethylidene)-1-(3-(ethoxycarbonyl)-4,5,6,7-tetrahydrobenzo[b]thiophene-2-yl)-4,5-dihydro-1H-pyrrole-3-carboxylic acid of formula 1:

.

EFFECT: obtaining a compound with high output, having pronounced antimicrobial activity against gram-positive microorganisms, as well as low toxicity.

1 cl, 1 tbl, 3 ex

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RU 2 738 405 C1

Authors

Shipilovskikh Sergej Aleksandrovich

Rubtsov Aleksandr Evgenevich

Makhmudov Ramiz Ragibovich

Tkachenko Aleksandr Georgievich

Nesterova Larisa Yurevna

Dates

2020-12-11Published

2020-05-26Filed