ANTIFIBROGENIC COMPOUNDS, METHODS AND USE THEREOF Russian patent published in 2020 - IPC A61K31/198 A61K31/47 A61P19/04 

Abstract RU 2726416 C2

FIELD: medicine; pharmaceuticals.

SUBSTANCE: group of inventions relates to the field and specifically to use of a compound of formula I: I, where E1 is H, OH or NH2; E2 is H, OH or NH2; E3 is H, OH or NH2; E4 is H, OH or NH2; A is H or NH2; D is ; or A and D form 6-member ring of formula: ; G is N; L1 is OH; for treating a fibrotic disease. Group of inventions also relates to a method of treating a fibrosing disease by administering said compounds; pharmaceutical composition containing said compounds, and commercial package containing said compositions.

EFFECT: group of inventions provides new agents and methods of treating fibrosis.

35 cl, 13 ex, 19 dwg

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RU 2 726 416 C2

Authors

Gakhari Aziz

Li Yunyuan

Kilani Rukhangiz T.

Khartvell Rajan

Dates

2020-07-14Published

2014-06-04Filed