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(19)

(11)

2 733 402

(13)

(51)

IPC

C07D417/14(2006-01-01)

C07D471/04(2006-01-01)

A61K31/424(2006-01-01)

A61K31/431(2006-01-01)

A61K31/439(2006-01-01)

A61P31/04(2006-01-01)

(21) (22)

Application

2018134948, 2017-03-02

(24)

Start date

2017-03-02

(22)

Actual filing date

2017-03-02

(45)

Published

2020-10-01

(72)

Inventor

Liu, WeiguoDing, Fa-XiangSun, WanyingDejesus, Reynalda, KehTang, HaifengHuang, XianhaiJian, JinlongGuo, YanWang, Hongwu

(73)

Holder

Merck Sharp Dohme Corp.

BICYCLIC ARYL MONOBACTAM COMPOUNDS AND METHODS OF USING SAID COMPOUNDS FOR TREATING BACTERIAL INFECTIONS Russian patent published in 2020 - IPC C07D417/14 C07D471/04 A61K31/424 A61K31/431 A61K31/439 A61P31/04

Abstract RU 2733402 C2

FIELD: pharmaceuticals.

SUBSTANCE: present invention relates to bicyclic aryl monobactam compounds listed in the patent claim, and pharmaceutically acceptable salts thereof, in particular trifluoroacetic salts, having antibacterial activity.

EFFECT: disclosed are bicyclic aryl monobactam compounds and methods of using them for treating bacterial infections.

4 cl, 9 tbl, 73 ex

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RU 2 733 402 C2

Authors

Liu, Weiguo

Ding, Fa-Xiang

Sun, Wanying

Dejesus, Reynalda, Keh

Tang, Haifeng

Huang, Xianhai

Jian, Jinlong

Guo, Yan

Wang, Hongwu

Dates

2020-10-01—Published

2017-03-02—Filed