Show metadata Hide metadata

(19)

(11)

2 733 402

(13)

(51)

IPC

C07D417/14(2006-01-01)

C07D471/04(2006-01-01)

A61K31/424(2006-01-01)

A61K31/431(2006-01-01)

A61K31/439(2006-01-01)

A61P31/04(2006-01-01)

(21) (22)

Application

2018134948, 2017-03-02

(24)

Start date

2017-03-02

(22)

Actual filing date

2017-03-02

(45)

Published

2020-10-01

(72)

Inventor

Liu, WeiguoDing, Fa-XiangSun, WanyingDejesus, Reynalda, KehTang, HaifengHuang, XianhaiJian, JinlongGuo, YanWang, Hongwu

(73)

Holder

Merck Sharp Dohme Corp.

BICYCLIC ARYL MONOBACTAM COMPOUNDS AND METHODS OF USING SAID COMPOUNDS FOR TREATING BACTERIAL INFECTIONS Russian patent published in 2020 - IPC C07D417/14 C07D471/04 A61K31/424 A61K31/431 A61K31/439 A61P31/04

Abstract RU 2733402 C2

FIELD: pharmaceuticals.

SUBSTANCE: present invention relates to bicyclic aryl monobactam compounds listed in the patent claim, and pharmaceutically acceptable salts thereof, in particular trifluoroacetic salts, having antibacterial activity.

EFFECT: disclosed are bicyclic aryl monobactam compounds and methods of using them for treating bacterial infections.

4 cl, 9 tbl, 73 ex

Similar patents RU2733402C2

Title	Year	Author	Number
BIARILE MONOBACTAM COMPOUNDS AND METHODS OF THEIR APPLICATION FOR TREATMENT OF BACTERIAL INFECTIONS	2016	Tang, Haifeng Liu, Weiguo Ding, Fa-Xiang Sun, Wanying Zang, Yi Pan, Weidong Ogawa, Anthony Brockunier, Linda Huang, Xianhai Wang, Hongwu Mal, Rudrajit Biftu, Tesfaye Park, Min Guo, Yan Jiang, Jinlong Chen, Helen Plummer, Christopher, W.	RU2746129C2
THERAPEUTIC COMPOUNDS AND COMPOSITIONS	2015	Chrusciel Robert A. Gadwood Robert C. Hayward Neil J. Melnick Michael J. Navia Manuel Poel Toni J. Stewart Catherine A. Stassen Frans L.	RU2733405C2
TETRASUBSTITUTED ALKENE COMPOUNDS AND USE THEREOF	2016	Bock, Mark Hao, Ming-Hong Korpal, Manav Nyavanandi, Vijay Kumar Puyang, Xiaoling Samajdar, Susanta Smith, Peter Gerard Wang, John Zheng, Guo Zhu Zhu, Ping	RU2733741C2
INHIBITOR CONTAINING BICYCLIC DERIVATIVE, METHOD OF PREPARATION AND USE THEREOF	2020	Su, Yidong Wang, Jun Bao, Rudi	RU2820948C2
COMPOUNDS	2016	Ding Xiao Jin Yun Liu Qian Ren Feng Sang Yingxia Stasi Luigi Piero Wan Zehong Wang Hailong Xing Weiqiang Zhan Yang Zhao Baowei	RU2725616C2
PYRUVATEKINASE MODULATORS AND THEIR USE	2018	Chianketta, Dzhovanni Kung, Charlz Lyu, Tao Padyana, Anil, Kumar Suj, Chzhikhua Tsaj, Chzhenvej Tsuj, Davej Tszi, Tszintszin	RU2797518C2
SUBSTITUTED BENZENE COMPOUNDS	2012	Kuntts Kevin Uejn Chesuort Richard Dunkan Kennet Uillyam Kajlkhak Khajke Varkholik Natali Klaus Kristin Natson Sara K. Vigl Timoti Dzhejms Nelson Seki Masasi	RU2629118C2
PIPERIDINYLPYRAZOLOPYRIMIDINONES AND USE THEREOF	2015	Ellermann Manuel Falot Gelle Kankho Grande Iolanda Khassfeld Jorma Kintsel Tom Kebberling Jokhannes Bajer Kristin Rerig Zuzanne Shpertsel Mikhael Shtampfuss Yan Majer Imke Kellnberger Maria Burkkhardt Nils Shlemmer Karl-Khajnts Shtegmann Kristian Shumakher Joakhim Verner Mattias Khajermann Jorg Khengeveld Villem Yan	RU2713937C2
PURINE COMPOUNDS INHIBITING PI3K, AND APPLICATION METHODS	2009	Kastanedo Zhorzhett Chukauri Irina Foulks Adrian Saterlin Daniel P. Van' Nan' Chi	RU2509081C2
PRIMARY CARBOXAMIDES AS BTK INHIBITORS	2014	Bonafu Dominik Devis Khiter M. Frenk Kristin E. Fridman Majkl M. Kherold Dzh. Martin Khoumann Majkl Z. Khantli Rejmond Osuma Ogastin Sheppard Dzhordzh Somal Gagandip K. Van Kamp Dzhennifer Van Epps Stejsi A. Vasudevan Anil Uollejs Grir A. Van Lu Van Lu Van Chzhi Uilson Noel S. Syuj Syandun	RU2708395C2

RU 2 733 402 C2

Authors

Liu, Weiguo

Ding, Fa-Xiang

Sun, Wanying

Dejesus, Reynalda, Keh

Tang, Haifeng

Huang, Xianhai

Jian, Jinlong

Guo, Yan

Wang, Hongwu

Dates

2020-10-01—Published

2017-03-02—Filed