5-ETHYL-4-METHYL-PYRAZOLE-3-CARBOXAMIDE DERIVATIVE HAVING TAAR AGONIST ACTIVITY Russian patent published in 2020 - IPC C07D413/12 A61K31/5377 A61P3/04 A61P3/06 A61P3/10 A61P9/00 A61P25/00 

Abstract RU 2731095 C2

FIELD: pharmaceuticals.

SUBSTANCE: invention relates to a compound of formula (I), which is 5-ethyl-4-methyl-N-[4-[(2S)morpholin-2-yl]phenyl]-1H-pyrazole-3-carboxamide, or to its pharmaceutically acceptable acid addition salt. Invention also relates to a method of producing a compound of formula (I), use thereof, a pharmaceutical composition, a method of activating TAAR.

EFFECT: obtaining a novel compound of formula (I) having TAAR agonist activity.

12 cl, 20 ex, 1 tbl

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RU 2 731 095 C2

Authors

Gallej Guido

Khener Marius

Norkross Rodzher

Pfliger Filipp

Dates

2020-08-28Published

2017-03-14Filed