4 - ((2-ARYL-2,4-DIHYDROXY-5-OXO-3-(3-OXO-3,4-DIHYDROQUINOXALIN-2-YL)-2,5-DIHYDRO-1N-PYRROL-1-YL)AMINO)BENZOIC ACIDS HAVING ANALGESIC ACTIVITY Russian patent published in 2020 - IPC C07D403/04 A61K31/4985 A61P29/00 

Abstract RU 2731215 C1

FIELD: chemistry.

SUBSTANCE: invention relates to 4-((2-aryl-2,4-dihydroxy-5-oxo-3-(3-oxo-3,4-dihydroquinoxalin-2-yl)-2,5-dihydro-1H-pyrrol-1-yl)amino)benzoic acids of the following general formula, where Ar = 4-Me-C6H4 (a) and Ar = 4-NO2-C6H4 (c).

EFFECT: compounds have analgesic activity.

1 cl, 1 tbl, 4 ex

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RU 2 731 215 C1

Authors

Mashevskaya Irina Vladimirovna

Makhmudov Ramiz Ragibovich

Prikhodko Yaroslav Igorevich

Dates

2020-08-31Published

2019-11-19Filed