ANTIMICROBIAL AGENT BASED ON 2-(R-AMINO-6-HYDROXY-7-(3-OXO-3,4-DIHYDROQUINOXALIN-2-yl)-7a-ARYLPYRROLO[2,1-b][1,3,4]THIADIAZOL-5(7aH)-ONES Russian patent published in 2024 - IPC C07D513/02 A61K31/407 A61K31/498 A61P31/04 

Abstract RU 2830076 C1

FIELD: chemistry.

SUBSTANCE: invention relates to biologically active compounds 2-(R1-amino-6-hydroxy-7-(3-oxo-3,4-dihydroquinoxalin-2-yl)-7a-arylpyrrolo[2,1-b][1,3,4]thiadiazol-5(7aH)-one of general formula (I), where R=H (a), CH3 (b); R1=CH2CH3 (a), H (b).

EFFECT: obtained compounds 2-(R1-amino-6-hydroxy-7-(3-oxo-3,4-dihydroquinoxalin-2-yl)-7a-arylpyrrolo[2,1-b][1,3,4]thiadiazole-5(7aH)-ones having antimicrobial activity.

1 cl, 1 tbl, 3 ex

(I)

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RU 2 830 076 C1

Authors

Mashevskaia Irina Vladimirovna

Belozerova Dzhamilia Nailevna

Balandina Svetlana Iurevna

Sukhanova Polina Vasilevna

Dates

2024-11-12Published

2024-03-17Filed