FIELD: organic chemistry.
SUBSTANCE: invention refers to benzodiazole compounds selected from: 1'-{[5-(aminomethyl)-1-(4,4,4-trifluorobutyl)-1H-1,3-benzodiazol-2-yl]methyl}-6'-fluoro-1', 2'-dihydrospiro[cyclopropane-1,3'-indol]-2'-one; 1'-((5-(aminomethyl)-1-(tetrahydro-2H-pyran-4-yl)-1H-benzo[d]imidazol-2-yl)methyl)-6'-fluoro-spiro[cyclopropane-1,3'-indoline]-2'-one and their pharmaceutically acceptable salts. What is also described is a pharmaceutical composition based on said compounds and a method of treating involving administering said compounds.
EFFECT: novel benzodiazole derivatives useful for treating or preventing an infection caused by respiratory-syncytial virus (RSV) are obtained.
3 cl, 6 tbl, 42 ex
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