HETEROCYCLIC SUBSTANCES-GPR119 AGONISTS Russian patent published in 2020 - IPC C07D417/14 A61K31/4535 A61K31/454 A61K31/506 A61P3/06 A61P5/50 

Abstract RU 2734500 C2

FIELD: medicine; pharmaceuticals.

SUBSTANCE: invention refers to compounds of formula (I) and use thereof for treating diseases and conditions mediated by GPR119. In general formula (I), each of X1, X2, X3, X4 and X5 independently represents N, S or CH; and X4 and X5 are combined with formation of five-member ring containing atom N, R1 and R2 are H, values A and B are given in the claim.

(I)

EFFECT: disclosed are heterocyclic substances—GPR119 agonists.

28 cl, 2 tbl, 40 ex

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RU 2 734 500 C2

Authors

Patil, Rakesh Ishwar

Verma, Jeevan

Kumar, Puneet

Gunjal, Amol, Pandurang

Rai, Himanshu

Rai, Santosh Kumar

Kumar, Anil

Dates

2020-10-19Published

2017-04-05Filed