NOVEL COMPOUNDS FOR INHIBITION OF JANUS KINASE 1 Russian patent published in 2025 - IPC C07D471/04 A61K31/437 A61P1/00 A61P17/06 A61P19/02 A61P35/00 

Abstract RU 2833828 C2

FIELD: pharmaceutics.

SUBSTANCE: present invention relates to novel selective Janus kinase 1 (JAK1) inhibitors, methods of producing said inhibitors, a pharmaceutical composition containing said inhibitors and use thereof.

EFFECT: development of new compounds as selective JAK1 inhibitors.

10 cl, 2 dwg, 4 tbl, 8 ex

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RU 2 833 828 C2

Authors

Rai, Santosh Kumar

Bandgar, Makhadev

Ali, Sazid

Rai, Khimanshu

Gundzhal, Amol Pandurang

Patil, Rakesh Isvar

Bapuram, Shrinivasa Reddi

Kumar, Anil

Dates

2025-01-29Published

2020-05-26Filed